ITC

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For a full dataset and details of experiment click on the datum link or any thermodynamic datum in the table below.

DatumProteinLigandΔG (kJ/mol)ΔH (kJ/mol)TΔS (kJ/mol)KD (µM)ΔCp (J/mol)
Link Trypsin Benzamidine-para-amide Benzamidine-para-amide diagram
Benzamidine-para-amide
-29.3 -24.1 5.2 5.95 -0.52
Link Trypsin Benzamidine-para-amide Benzamidine-para-amide diagram
Benzamidine-para-amide
-29.1 -26.9 2.2 7.87 -0.52
Link Trypsin Benzamidine-para-amide Benzamidine-para-amide diagram
Benzamidine-para-amide
-29.1 -30.2 -1.4 9.71 -0.52
Link Trypsin Benzamidine-para-amide Benzamidine-para-amide diagram
Benzamidine-para-amide
-28.8 -33.0 -4.2 14.08 -0.52