For a full dataset and details of experiment click on the datum link or any thermodynamic datum in the table below.
Datum | Protein | Ligand | ΔG (kJ/mol) | ΔH (kJ/mol) | TΔS (kJ/mol) | KD (µM) | ΔCp (J/mol) |
Link |
Disabled Homolog 1 (H81Q)
|
D-myo-inositol-1,4,5-triphosphate
 D-myo-inositol-1,4,5-triphosphate
|
-26.78
|
-41.0
|
-14.23
|
18.0
|
|
Link |
Disabled Homolog 1 (H81Q)
|
TKSMNFDNPVYRKT
 TKSMNFDNPVYRKT
|
-33.05
|
-45.19
|
-12.13
|
1.6
|
|
Link |
Disabled Homolog 1 (K45A)
|
TKSMNFDNPVYRKT
 TKSMNFDNPVYRKT
|
-32.22
|
-42.26
|
-10.04
|
2.3
|
|
Link |
Disabled Homolog 1 (K45A/K82A)
|
TKSMNFDNPVYRKT
 TKSMNFDNPVYRKT
|
-31.38
|
-36.82
|
-5.44
|
3.0
|
|
Link |
Disabled Homolog 1 (K45E)
|
TKSMNFDNPVYRKT
 TKSMNFDNPVYRKT
|
-32.22
|
-44.35
|
-12.13
|
2.2
|
|
Link |
Disabled Homolog 1 (K45E/K82Q)
|
TKSMNFDNPVYRKT
 TKSMNFDNPVYRKT
|
-32.22
|
-42.68
|
-10.46
|
2.1
|
|
Link |
Disabled Homolog 1 (K45Q)
|
TKSMNFDNPVYRKT
 TKSMNFDNPVYRKT
|
-31.38
|
-33.89
|
-2.51
|
2.9
|
|
Link |
Disabled Homolog 1 (K45Q/K82Q)
|
TKSMNFDNPVYRKT
 TKSMNFDNPVYRKT
|
-31.8
|
-38.91
|
-7.11
|
2.7
|
|
Link |
Disabled Homolog 1 (K82A)
|
TKSMNFDNPVYRKT
 TKSMNFDNPVYRKT
|
-33.47
|
-46.02
|
-12.55
|
1.4
|
|
Link |
Disabled Homolog 1 (K82Q)
|
TKSMNFDNPVYRKT
 TKSMNFDNPVYRKT
|
-33.05
|
-60.67
|
-27.61
|
1.7
|
|
Link |
Disabled Homolog 1 (S114Y)
|
D-myo-inositol-1,4,5-triphosphate
 D-myo-inositol-1,4,5-triphosphate
|
-33.89
|
-102.09
|
-68.2
|
1.2
|
|
Link |
Disabled Homolog 1 (native)
|
D-myo-inositol-1,4,5-triphosphate
 D-myo-inositol-1,4,5-triphosphate
|
-33.89
|
-80.33
|
-46.44
|
1.2
|
|
Link |
Disabled Homolog 1 (native)
|
TKSMNFDNPVYRKT
 TKSMNFDNPVYRKT
|
-32.22
|
-40.17
|
-7.95
|
3.0
|
|
Link |
Endo-1,4-Beta Glucanase EngF
|
Cellohexaose
 Cellohexaose
|
-27.22
|
-60.81
|
-33.59
|
17.01
|
-0.61
|
Link |
Endo-1,4-Beta Glucanase EngF
|
Cellopentaose
 Cellopentaose
|
-24.25
|
-68.38
|
-44.13
|
56.5
|
-0.8
|
Link |
Endo-1,4-Beta Glucanase EngF
|
Cellotetraose
 Cellotetraose
|
-17.53
|
-74.59
|
-57.06
|
833.33
|
|
Link |
Endo-1,4-Beta Glucanase EngF (D54A)
|
Cellohexaose
 Cellohexaose
|
-22.02
|
-51.63
|
-29.61
|
138.89
|
-0.53
|
Link |
Endo-1,4-Beta Glucanase EngF (N137A)
|
Cellohexaose
 Cellohexaose
|
-20.32
|
-53.43
|
-33.11
|
277.78
|
-0.88
|
Link |
Endo-1,4-Beta Glucanase EngF (N52A)
|
Cellohexaose
 Cellohexaose
|
-21.24
|
-51.76
|
-30.52
|
188.68
|
-0.68
|
Link |
Endo-1,4-Beta Glucanase EngF (R92A)
|
Cellohexaose
 Cellohexaose
|
-20.16
|
-61.97
|
-41.81
|
294.12
|
-0.99
|